Tadalafil entfaltet seine Wirkung über eine selektive Hemmung der PDE5, wodurch die Konzentration von cGMP im glatten Muskelgewebe stabil bleibt. Diese biochemische Modulation resultiert in einer langanhaltenden Relaxation der Gefäßwände. Der Wirkstoff wird nach oraler Einnahme effizient resorbiert, mit einer Bioverfügbarkeit von rund 80 %. Seine Halbwertszeit von bis zu 36 Stunden ist innerhalb dieser Substanzklasse außergewöhnlich. Abgebaut wird er in der Leber, hauptsächlich durch CYP3A4, mit anschließender biliärer Exkretion. Typische unerwünschte Wirkungen entstehen durch eine verstärkte Vasodilatation, etwa Kopfschmerzen oder Flush. Pharmakologisch wird cialis generika vor allem durch die verlängerte Wirkungsdauer charakterisiert.
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OKTOBER 2005
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Tratamiento con antihipertensivos y función cognitiva en la enfermedad de Alzheimer Profesor Ingmar Skoog, M.D., Ph.D. Unidad de Epidemiología Neuropsiquiátrica, Instituto de Neurociencia y Fisiología, Sahlgrenska Academy, Universidad de Gotemburgo, Suecia Se ha demostrado que el tratamiento de la hipertensión reduce considerablemente el riesgo cardiovascular pero, entre
VOLUNTARY SECTOR Introduction Voluntarism is an integral part of Indian society and dates back to ancient times when it operated in the fields of education, medicine, cultural promotion, and in crises such as droughts and famines. Modern indigenous forms of voluntary organisations began to appear in the colonial period. According to the World Development Report (World Bank, 1993),"
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